XVIII - Antivirals Flashcards Preview

Pharmacology > XVIII - Antivirals > Flashcards

Flashcards in XVIII - Antivirals Deck (13)
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1
Q

Guanosine analogue, treatment of HSV and VZV, requires activation by viral thymidine kinase, SE: crystalluria

A

Acyclovir

2
Q

Treatment of CMV, requires activation by viral thymidine kinase

A

Gancyclovir

3
Q

Pyrophosphate analogue, treatment of HSV, VZV and CMV, does not require activation by viral thymidine kinase

A

Foscarnet

4
Q

Prevents viral uncoating, Influenza A, Rubella, SE: cerebellar dysfunction, livedo reticularis

A

Amantadine

5
Q

Neuraminidase inhibitor, DOC for Influenza

A

Oseltamivir

6
Q

Treatment for Hepatitis B

A

Lamivudine

7
Q

Treatment for Hepatitis C and RSV

A

Ribavirin

8
Q

Nucleoside reverse transcriptase inhibitor (NRTI), requires phosphorylation, primary drug for HIV, prevents vertical transmission of HIV, SE: lactic acidosis

A

Zidovudine (AZT)

9
Q

Non-nucleoside reverse transcriptase inhibitor (NNRTI), no phosphorylation required, SE: hepatotoxic

A

Delavirdine

10
Q

Protease inhibitor, SE: fat redistribution syndrome, hyperlipidemia, insulin resistance

A

Indinavir

11
Q

Fusion inhibitor, binds gp41 subunit

A

Enfuvirtide

12
Q

Binding inhibitor, CCR5 antagonist

A

Maraviroc

13
Q

Non-Nucleoside Reverse Transcriptase Inhibitors

A

Nevirapine, Efavirenz, Delavirdine